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Sapunaric Frédéric

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Main Referenced Co-authors
Frère, Jean-Marie  (3)
Levy, Stuart B. (3)
Amoroso, Ana Maria  (2)
Colau, Didier (2)
Colette, Delphine (2)
Main Referenced Keywords
Tetracycline (4); Efflux (3); Resistance (3); Anti-Bacterial Agents/pharmacology (1); Antimicrobial Resistance (1);
Main Referenced Unit & Research Centers
CIP - Centre d'Ingénierie des Protéines - ULiège [BE] (2)
Center for Adaptation Genetics and Drug Resistance (2)
Main Referenced Disciplines
Microbiology (8)
Oncology (2)
Biochemistry, biophysics & molecular biology (1)

Publications (total 11)

The most downloaded
801 downloads
Dolusic, E., Larrieu, P., Blanc, S., Sapunaric, F., Pouyez, J., Moineaux, L., Colette, D., Stroobant, V., Pilotte, L., Colau, D., Ferain, T., Fraser, G., Galleni, M., Frère, J.-M., Masereel, B., Van den Eynde, B., Wouters, J., & Frederick, R. (2011). Discovery and preliminary SARs of keto-indoles as novel indoleamine 2,3-dioxygenase (IDO) inhibitors. European Journal of Medicinal Chemistry, 46 (7), 3058-65. doi:10.1016/j.ejmech.2011.02.049 https://hdl.handle.net/2268/92049

The most cited

58 citations (Scopus®)

Dolusic, E., Larrieu, P., Blanc, S., Sapunaric, F., Pouyez, J., Moineaux, L., Colette, D., Stroobant, V., Pilotte, L., Colau, D., Ferain, T., Fraser, G., Galleni, M., Frère, J.-M., Masereel, B., Van den Eynde, B., Wouters, J., & Frederick, R. (2011). Discovery and preliminary SARs of keto-indoles as novel indoleamine 2,3-dioxygenase (IDO) inhibitors. European Journal of Medicinal Chemistry, 46 (7), 3058-65. doi:10.1016/j.ejmech.2011.02.049 https://hdl.handle.net/2268/92049

Dolusic, E., Larrieu, P., Blanc, S., Sapunaric, F., Pouyez, J., Moineaux, L., Colette, D., Stroobant, V., Pilotte, L., Colau, D., Ferain, T., Fraser, G., Galleni, M., Frère, J.-M., Masereel, B., Van den Eynde, B., Wouters, J., & Frederick, R. (2011). Discovery and preliminary SARs of keto-indoles as novel indoleamine 2,3-dioxygenase (IDO) inhibitors. European Journal of Medicinal Chemistry, 46 (7), 3058-65. doi:10.1016/j.ejmech.2011.02.049
Peer Reviewed verified by ORBi

Dolusic, E., Larrieu, P., Blanc, S., Sapunaric, F., Norberg, B., Moineaux, L., Colette, D., Stroobant, V., Pilotte, L., Colau, D., Ferain, T., Fraser, G., Galleni, M., Frère, J.-M., Masereel, B., Van den Eynde, B., Wouters, J., & Frederick, R. (2011). Indol-2-yl ethanones as novel indoleamine 2,3-dioxygenase (IDO) inhibitors. Bioorganic and Medicinal Chemistry, 19 (4), 1550-61. doi:10.1016/j.bmc.2010.12.032
Peer Reviewed verified by ORBi

Sapunaric, F., & Levy, S. B. (2007). Interdomain loop mutation Asp190Cys of the tetracycline efflux transporter TetA(B) decreases affinity for substrate. Antimicrobial Agents and Chemotherapy. doi:10.1128/AAC.00357-07
Peer Reviewed verified by ORBi

Fraipont, C., Sapunaric, F., Zervosen, A., Auger, G., Devreese, B., Lioux, T., Blanot, D., Mengin-Lecreulx, D., Herdewijn, P., Van Beeumen, J., Frère, J.-M., & Nguyen-Distèche, M. (28 March 2006). Glycosyl transferase activity of the Escherichia coli penicillin-binding protein 1b: Specificity profile for the substrate. Biochemistry, 45 (12), 4007-4013. doi:10.1021/bi051055m
Peer Reviewed verified by ORBi

Sapunaric, F., & Levy, S. B. (July 2005). Substitutions in the interdomain loop of the Tn10 TetA efflux transporter alter tetracycline resistance and substrate specificity. Microbiology, 151, 2315-2322. doi:10.1099/mic.0.27997-0
Peer Reviewed verified by ORBi

Sapunaric, F., Aldema-Ramos, M., & McMurry, L. M. (2005). Tetracycline resistance: Efflux, Mutations and, Other Mechanisms. In D. G. White, M. N. Alekshun, ... P. F. McDermott, Frontiers in Antimicrobial Resistance: A Tribute to Stuart B. Levy (pp. 1: 3-18). Washington, United States: ASM Press.

Sapunaric, F., & Levy, S. B. (August 2003). Second-site suppressor mutations for the serine 202 to phenylalanine substitution within the interdomain loop of the tetracycline efflux protein Tet(C). Journal of Biological Chemistry, 278, 28588–28592. doi:10.1074/jbc.M302658200
Peer Reviewed verified by ORBi

Sapunaric, F., Franssen, C., Stefanic, P., Amoroso, A. M., Dardenne, O., & Coyette, J. (2003). Redefining the role of psr in beta-lactam resistance and cell autolysis of Enterococcus hirae. Journal of Bacteriology, 185 (20), 5925-35. doi:10.1128/JB.185.20.5925-5935.2003
Peer Reviewed verified by ORBi

Sapunaric, F. (2002). Rôle régulateur de la protéine Psr sur la synthèse de la protéine PBP5 impliquée dans la résistance d'Enterococcus hirae aux beta-lactamines : Mythe ou réalité ? [Doctoral thesis, ULiège - Université de Liège]. ORBi-University of Liège. https://orbi.uliege.be/handle/2268/92271

Duez, C., Zorzi, W., Sapunaric, F., Amoroso, A. M., Thamm, I., & Coyette, J. (September 2001). The Penicillin Resistance of Enterococcus Faecalis Jh2-2r Results from an Overproduction of the Low-Affinity Penicillin-Binding Protein Pbp4 and Does Not Involve a Psr-Like Gene. Microbiology, 147 (Pt 9), 2561-9. doi:10.1099/00221287-147-9-2561
Peer Reviewed verified by ORBi

Duez, C., Thamm, I., Sapunaric, F., Coyette, J., & Ghuysen, J.-M. (1998). The Division and Cell Wall Gene Cluster of Enterococcus Hirae S185. DNA Sequence: the Journal of DNA Sequencing and Mapping, 9 (3), 149-161. doi:10.3109/10425179809072190
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